Our inaugural half-day symposium brought together around 100 academic and industrial scientists as well as PhD students, and featured a keynote lecture by Stuart Conway from the University of Oxford (UK). It provided ample opportunities for networking, a poster session, and a reception at the end of the day.
Program
13.00-13.05 Welcome (Trond Ulven)
13.05-14.00 Stuart Conway (Univ. of Oxford)
Internal hydrogen bonds in the design of CREBBP bromodomain ligands
14.00-14.30 Luigi Piero Stasi (Nuevolution)
DNA Encoded Library Technology: From hits to clinical candidates
14.30-15.00 Coffee break
15.00-15.45 Young investigators (nominees for the EFMC YI prize)
Nima Rajabi
Developing Mechanism-based Inhibitors of the Human Sirtuin 5 Deacylase
Jorge Peiró
Reactive oxygen species sensitive prodrugs for the treatment of chronic inflammatory diseases
15.45-16.15 Thomas B. Poulsen (AU)
Natural products guiding the search for new therapeutic targets
16.15-16.45 Coffee break
16.45-17.15 Daniel Greve (LEO Pharma)
Discovery of Janus kinase inhibitors for topical treatment of psoriasis
17.15-17.45 Jesper Langgaard Kristensen (KU) Inaugural lecture:
Development of selective Serotonin 2A receptor agonists
17.45-17.50 EFMC YI winner announced
17.50-19.00 Reception and poster session
Posters
- Kaja Borup Løvschall, Alexander N. Zelikin
Macromolecular (pro) drugs as broad-spectrum antiviral agents - Raoul Walther, Signe M. Nielsen, Rikke Christiansen, Rikke Louise Meyer, Alexander N. Zelikin
Self-immolative linkers pave the way to fluoroquinolone glucuronide produgs: A proof of concept study to treat implant associated biofilms - Camilla Kaas Frich,Alexander N. Zelikin
Albumin-polymer-drug conjugates: Combination therapy with extended circulation time - Nima Rajabi, Marina Auth, Kathrin R. Troelsen, Martin Pannek, Martin Fontenas, Clemens Steegborn, Andreas S. Madsen, and Christian A. Olsen
Mechanism-based inhibitors of the human sirtuin 5 deacylase - Mads Holmgaard Kaspersen, Christoffer Vogsen Heidtmann, Laura Jenkins, Julia Dunlop, Graeme Milligan and Trond Ulven
Synthesis and in vitro evaluation of hydroxyfatty acids and synthetic analogues on GPR84
Venue
Auditorium A4
Dept. of Drug Design and Pharmacology
University of Copenhagen
Universitetsparken 2
2100 Copenhagen